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KIT kinase domain mutant D816H in complex with sunitinib
Autogenerated by
for
Millhill
Created on Mon, 2020-12-21 17:01, last updated on Mon, 2020-12-21 17:01
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General Information
This Model was autogenerated from the
"Quick Submit"
tool.
Model ID
3DPX-015291
Category
Proteins, Macromolecules and Viruses
Keyword(s)
KIT Kinase domain, Sutent binding, drug resistance, ATP-binding, Disease mutation, glycoprotein, Immunoglobulin Domain, KINASE, Membrane, Nucleotide-binding
Protein Data Bank ID
3G0F
Experimental Method
X-RAY DIFFRACTION
Resolution
2.6
Model Details
Associated Species
Spodoptera frugiperda
Oligomeric Details
tetrameric
R-Factor
0.207
Scattering Type
x-ray
Attribution
PubMed ID
19 164 557
Digital Object Identifier (DOI)
10.1073/pnas.0812413106
Citation Title
KIT kinase mutants show unique mechanisms of drug resistance to imatinib and sunitinib in gastrointestinal stromal tumor patients.
Citation Year
2009
STL/VRML Files
PDB-3G0F-ribbon-secondary.wrl
PDB-3G0F-ribbon-rainbow.wrl
PDB-3G0F-ribbon-bychain.wrl
PDB-3G0F-ribbon.stl
PDB-3G0F-surf-bychain.wrl
PDB-3G0F-surf-hydropathy.wrl
PDB-3G0F-surf-coulombic.wrl
PDB-3G0F-surf.stl
PDB-3G0F.zip
X3D Files
PDB-3G0F-ribbon-secondary.x3d
PDB-3G0F-ribbon-rainbow.x3d
PDB-3G0F-ribbon-bychain.x3d
PDB-3G0F-ribbon.x3d
PDB-3G0F-surf-bychain.x3d
PDB-3G0F-surf-hydropathy.x3d
PDB-3G0F-surf-coulombic.x3d
PDB-3G0F-surf.x3d
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